| Cat.No.: | BSM-0252 |
| Product Name: | UNC1999 |
| CAS No.: | 1431612-23-5 |
| Figure: |
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| Synonyms: | N-{(6-methyl-2-oxo-4-propyl-1H-pyridin-3-yl)methyl}-1-propan-2-yl-6-{6-(4-propan-2-ylpiperazin-1-yl)pyridin-3-yl}indazole-4-carboxamide |
| Description: | A potent histone H3-lysine 27 (H3K27) methyltransferase EZH2 inhibitor (IC50 = 2 nM). It suppresses global H3K27 trimethylation/demethylation and inhibits the growth of mixed lineage leukemia (MLL)-rearranged leukemia cells. |
| Appearance: | White to off-white solid |
| Molecular Weight: | 569.74 |
| Purity: | ≥98% by HPLC |
| Storage: | -20°C |
| Targets: | EZH1; EZH2 |
| Molecular Formula: | C33H43N7O2 |
| MDL Number: | MFCD17215972 |
| Solubility: | DMSO (~15 mg/ml) |
| Shipping Conditions: | Gel Pack |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Bioactive Small Molecules | ||
| BSM-0006 | GSK343 | Inquiry |
| BSM-0059 | 3-Deazaneplanocin A | Inquiry |
| BSM-0060 | 3-Deazaneplanocin A hydrochloride | Inquiry |
| ◆ Extracts & Lysates | ||
| EL-0024 | Recombinant Human EZH1 293 Cell Lysate | Inquiry |
| EL-0025 | Recombinant Human EZH2 293 Cell Lysate | Inquiry |
| Related Gene / Proteins | |||
| ezh1 | EZH2 | ||
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