| Cat.No.: | BSM-0214 |
| CAS No.: | 1613695-14-9 |
| Figure: |
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| Synonyms: | 2-[2-(3-Chloro-4-methoxyphenyl)ethyl]-5-(dimethyl-1,2-oxazol-4-yl)-1-[(2S)-2-(morpholin-4-yl)propyl]-1H-1,3-benzodiazole |
| Description: | SGC-CBP30 is a potent and selective CREBBP/EP300 bromodomain inhibitor with IC values of 21-69 and 38 nM for CREBBP and EP300 bromodomains, respectively. SGC-CBP30 has little activity against other bromodomains at concentrations up to 1 mM. |
| Appearance: | Off-white solid |
| Molecular Weight: | 509.04 |
| Purity: | ≥98% by HPLC |
| Storage: | -20°C |
| Targets: | CREBBP/EP300 bromodomin |
| Molecular Formula: | C28H33ClN4O3 |
| MDL Number: | MFCD00386477 |
| Solubility: | DMSO (>30 mg/ml) |
| Shipping Conditions: | Gel Pack |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Bioactive Small Molecules | ||
| BSM-0038 | CTPB | Inquiry |
| BSM-0073 | Anacardic Acid | Inquiry |
| BSM-0094 | C646 | Inquiry |
| ◆ Cell Lines | ||
| CL-0055 | Human CREBBP Knockout Cell Line 1bp insertion | Inquiry |
| CL-0061 | Human EP300 Knockout Cell Line 13bp deletion | Inquiry |
| Related Gene / Proteins | |||
| CREB | CREB3 | crebbp | CRISP1 |
| CRISP3 | CRP | EP300 | EPC1 |
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