| Cat.No.: | BSM-0105 |
| Product Name: | CPI-203 |
| CAS No.: | 1446144-04-2 |
| Figure: |
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| Synonyms: | (6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide |
| Description: | CPI-203 is an analog of (+)-JQ1. Acts as a BET bromodomain inhibitor. It is comparable or superior to (+)-JQ1 in inhibiting BRD4 binding and action in vitro or in cells.CPI-203 arrests the growth of leukemic T cells in vitro (EC₅₀ = 91 nM) and rapidly suppresses leukemia burden in mice. |
| Appearance: | White solid |
| Molecular Weight: | 399.9 |
| Purity: | ≥98% by HPLC |
| Storage: | -20°C |
| Targets: | BET bromodomain |
| Molecular Formula: | C₁₉H₁₈ClN₅OS |
| MDL Number: | MFCD00866266 |
| Solubility: | DMSO (>35 mg/ml) |
| Shipping Conditions: | Gel Pack |
| Warning: | For Research Use Only! Not For Use in Humans. |
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