| Cat.No.: | BSM-0087 |
| CAS No.: | 1883429-22-8 |
| Figure: |
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| Synonyms: | 4-(4-((dimethylamino)methyl)-2,5-dimethoxyphenyl)-2-methyl-2,7-naphthyridin-1(2H)-one |
| Description: | BI-9564 is a potent, selective and cell-permeable BRD9 and BRD7 inhibitor (Kd values are 14 and 239 nM, respectively). Displays selectivity for BRD9/7 over 48 other bromodomains, 324 kinases and 55 GPCRs. Inhibits proliferation of AML cell lines in vitro and reduces AML tumor xenograft growth in vivo. |
| Appearance: | Crystalline solid |
| Molecular Weight: | 353.41 |
| Purity: | ≥98% by HPLC |
| Storage: | -20°C |
| Targets: | BRD9 and BRD7 |
| Molecular Formula: | C₂₀H₂₃N₃O₃ |
| MDL Number: | MFCD16038904 |
| Solubility: | DMSO |
| Shipping Conditions: | Gel Pack |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Synthetic Peptides | ||
| SP-0001 | Bromodomain Non-Acetylated Ligand 4 | Inquiry |
| SP-0002 | Bromodomain Non-Acetylated Ligand 3 | Inquiry |
| SP-0003 | Bromodomain Non-Acetylated Ligand 1 | Inquiry |
| SP-0004 | Bromodomain Ligand 3 | Inquiry |
| SP-0006 | Bromodomain Ligand 4 | Inquiry |
| Related Gene / Proteins | |||
| BRCA1 | BRCA2 | BRCC3 | BRD |
| brd1 | brd2 | brd3 | brd4 |
| BRD7 | BRD8 | brd9 | brdt |
| BRL | BRM | BRMS1 | BRPF1 |
| BRPF2 | brpf3 | BRWD1 | BRWD3 |
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