| Cat.No.: | BSM-0030 |
| Product Name: | PF-06405761 |
| CAS No.: | 1403764-72-6 |
| Abbr: | PF-06405761(BRD4) |
| Synonyms: | CAP, HUNK1, HUNKI, MCAP |
| Description: | PF-06405761 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM. |
| Molecular Weight: | 347.39 |
| Purity: | > 95% |
| Storage: | 4°C |
| Targets: | BRD4 |
| IC50: | 0.22 μM |
| Molecular Formula: | C16H17N3O4S |
| Chemical Name: | 2-methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide |
| Warning: | For Research Use Only! Not For Use in Humans. |
| Product Types | ||
| ◆ Synthetic Peptides | ||
| SP-0001 | Bromodomain Non-Acetylated Ligand 4 | Inquiry |
| SP-0002 | Bromodomain Non-Acetylated Ligand 3 | Inquiry |
| SP-0003 | Bromodomain Non-Acetylated Ligand 1 | Inquiry |
| SP-0004 | Bromodomain Ligand 3 | Inquiry |
| SP-0006 | Bromodomain Ligand 4 | Inquiry |
| Related Gene / Proteins | |||
| BRCA1 | BRCA2 | BRCC3 | BRD |
| brd1 | brd2 | brd3 | brd4 |
| BRD7 | BRD8 | brd9 | brdt |
| BRL | BRM | BRMS1 | BRPF1 |
| BRPF2 | brpf3 | BRWD1 | BRWD3 |
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